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. 2006 Jun 29;575(Pt 1):5–10. doi: 10.1113/jphysiol.2006.111203

Table 1.

Cleavage products of amyloid precursor protein (APP) and their suggested physiological roles

Peptide Cleavage process Known function Reference
sAPPα α-secretase cleavage of APP Neuroprotective? Involved in blood clotting? Smith et al. 1990
Up-regulates BKCa activity Furukawa et al. 1996
C83 α-secretase cleavage of APP None known, but may be associated with neurodegeneration Rockenstein et al. 2005
p3 γ-secretase cleavage of C83 None known? Pardossi-Piquard et al. 2005
AICD/CFTγ γ-secretase cleavage of C83 Transcriptional regulation (e.g. of neprylisin) Leissring et al. 2002
sAPPβ β-secretase cleavage of APP Neuroprotective?
C99 β-secretase cleavage of APP Altered acetylcholinesterase activity and behavioural influences Dumont et al. 2005
γ-secretase cleavage of Depress synaptic activity Kamenetz et al. 2003
β-secretase cleaved of APP Regulation of Kv expression Ramsden et al. 2001; Plant et al. 2005
Regulation of Cav Ramsden et al. 2002